70.具有tetrahydrodiazepine結構的抗癌藥為:
(A)Cytarabine
(B)Pentostatin
(C)Paclitaxel
(D)Teniposide
答案:登入後查看
統計: A(587), B(1512), C(658), D(615), E(0) #416824
統計: A(587), B(1512), C(658), D(615), E(0) #416824
詳解 (共 9 筆)
#1098984
(A)Cytarabine 屬於cytidine analog + arabinose (B)Pentostatin 具有tetrahydrodiazepine
+ imidazole (C)Paclitaxel 屬於ditepenoids(二萜類),具有taxane
(D)Teniposide 屬於epipodophyllotoxins,具有lignan
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2
#1243746
79.抗癌藥pentostatin為下列何種酵素之抑制劑?
(A)Adenosine deaminase
(B)Thymidylate synthetase
(C)Dihydrofolate reductase
(D)Topoisomerase II
答案:A
(A)Adenosine deaminase
(B)Thymidylate synthetase
(C)Dihydrofolate reductase
(D)Topoisomerase II
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2
#1587025
Pentostatin雖有statin結尾,但不是抗血脂類
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2
#4909417
補充:adenosine相關藥物
抗癌=> pentostatin:adenosine deaminase inhibitor
抗病毒=> vidarabine(Ara-A):adenosine deaminase inhibitor
抗凝血=> dipyridamole:adenosine reuptake inhibitor(使adenosine太多)
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0
#853041
"Tetrahydrodiazepine" MOA- inhibition of adenosine deaminase

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#4838833
看到statin還以為是降血脂藥嗎? 其實是抗癌藥物啦! suprise! MDFK!
騙倒你了吧~ pentostatin
MOA inhibitor of adenosine deaminase
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0