39 下列何種抗黴菌藥物的代謝物可抑制 thymidylate synthetase,進而干擾 RNA 及蛋白質之生合成?
(A) Amphotericin B
(B) Ketoconazole
(C) Flucytosine
(D) Griseofulvin
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統計: A(15), B(22), C(172), D(24), E(0) #412818
統計: A(15), B(22), C(172), D(24), E(0) #412818
詳解 (共 3 筆)
#1616307
(A) Amphotericin B 影響細胞膜通透性,結合並且破壞ergosterol
(B) Ketoconazole 影響細胞膜通透性,抑制14-alpha-steroid demethylase,抑制ergosterol合成
(C) Flucytosine 5-FC,抑制DNA合成,抑制thymidylate synthetase
(D) Griseofulvin 抑制細胞分裂(有絲分裂)干擾微管聚合
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#841617
Flucytosine, or 5-fluorocytosine, a fluorinated pyrimidine analogue, is a synthetic antimycotic drug.
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