10.下列何種降血脂藥物之結構屬於isopropyl ester,口服後於小腸水解為活性代謝產物?
(A)Fenofibrate
(B)Ezetimibe
(C)Atorvastatin
(D)Cholestyramine
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統計: A(2802), B(1217), C(788), D(272), E(0) #624415
統計: A(2802), B(1217), C(788), D(272), E(0) #624415
詳解 (共 10 筆)
#2289294
給四樓,Fibrate 類藥物中Prodrug 只有 Clofibrate、Fenofibrate
剩下的ate結尾不是前驅藥喔
180
2
#1423396
33 下列何者屬於前驅藥物? (A) Gemfibrozil (B) Fenofibrate (C) Cholestyramine (D) Colestipol |
95
3
#2913073
補充:Statin類藥物裡面,Simuvastatin和Lovastatin也是Prodrug
43
1
#1025838
Fenofibrate (prodrug) ----> Fenofibric acid (active metabolite)
37
0
#1025835
32
1
#1603127
-ate. 前驅藥結尾
25
23
#3750031
Pro級的 功夫CF
就是clofibrate 和fenofibrate 是prodrug
16
1