22 下列那一種降壓藥物口服後最易被乙醯化(acetylation),而減少其藥效與生體可用率?
(A) Reserpine
(B) Clonidine
(C) Hydralazine
(D) Prazosin
答案:登入後查看
統計: A(242), B(317), C(1904), D(142), E(0) #417336
統計: A(242), B(317), C(1904), D(142), E(0) #417336
詳解 (共 5 筆)
#1416629
(C)Hydralazine
ADR:slow acetylation的人易造成Lupus erythematosus(紅斑性狼瘡)
ADR:slow acetylation的人易造成Lupus erythematosus(紅斑性狼瘡)
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#4661293
易被乙烯化的藥物:
1.primary aromatic amine:PAS (para-amino salicylic acid)
2.sulfonamide: sulfamethoxazole
3.hydrazine 和hydrazide:hydralazine、isoniazid
4.primary aliphatic amine: histamine
來源:阿摩前輩大大,非常感謝 ><
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